Grazioso Giovanni

Associate Professor
SSD
CHIM/08 - PHARMACEUTICAL CHEMISTRY
Competition sector
03/D1 - MEDICINAL, TOXICOLOGICAL AND NUTRITIONAL CHEMISTRY AND APPLIED TECHNOLOGIES

Contacts

Workplace

Via Mangiagalli, 25
20133 MILANO (MI)

Office phone number
02503 19352
Additional phone numbers
0250319351
University email address
Friday 10.30 -12.30, fixing an appointment by email
Reception office
Office 2015 - Lab. 2053 - Via Mangiagalli 25

Education

Research

Publications
  • Computationally Driven Structure Optimization, Synthesis, and Biological Evaluation of Imidazole-Based Proprotein Convertase Subtilisin/Kexin 9 (PCSK9) Inhibitors / C. Lammi, J. Sgrignani, A. Arnoldi, G. Lesma, C. Spatti, A. Silvani, G. Grazioso. - In: JOURNAL OF MEDICINAL CHEMISTRY. - ISSN 0022-2623. - 62:13(2019 Jun 18), pp. 6163-6174.
  • Rational design of allosteric modulators of the aromatase enzyme: An unprecedented therapeutic strategy to fight breast cancer / A. Spinello, S. Martini, F. Berti, M. Pennati, M. Pavlin, J. Sgrignani, G. Grazioso, G. Colombo, N. Zaffaroni, A. Magistrato. - In: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. - ISSN 0223-5234. - 168(2019 Apr 15), pp. 253-262.
  • Biological Characterization of Computationally Designed Analogs of peptide TVFTSWEEYLDWV (Pep2-8) with Increased PCSK9 Antagonistic Activity / C. Lammi, J. Sgrignani, A. Arnoldi, G. Grazioso. - In: SCIENTIFIC REPORTS. - ISSN 2045-2322. - 9:1(2019 Feb 20).
  • Oxidation State Dependent Conformational Changes of HMGB1 Regulate the Formation of the CXCL12/HMGB1 Heterocomplex / E.M.A. Fassi, J. Sgrignani, G. D'Agostino, V. Cecchinato, M. Garofalo, G. Grazioso, M. Uguccioni, A. Cavalli. - In: COMPUTATIONAL AND STRUCTURAL BIOTECHNOLOGY JOURNAL. - ISSN 2001-0370. - 17(2019), pp. 886-894.
  • Learning to Rank Food Images / D. Allegra, D. Erba, G.M. Farinella, G. Grazioso, P.D. Maci, F. Stanco, V. Tomaselli (LECTURE NOTES IN ARTIFICIAL INTELLIGENCE). - In: Image Analysis and Processing – ICIAP 2019 / [a cura di] E. Ricci, S. Rota Bulò, C. Snoek, O. Lanz, S. Messelodi, N. Sebe. - Prima edizione. - [s.l] : Springer Nature, 2019. - ISBN 9783030306441. - pp. 629-639 (( Intervento presentato al 20. convegno International Conference on Image Analysis and Processing tenutosi a Trento nel 2019.